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- 品牌：MedKoo
- 产地：美国
- 货号：407399
- cas：1202580-59-3
- 发布日期： 2022-07-20
- 更新日期： 2024-08-12
| 产地 | 美国 |
| 品牌 | MedKoo |
| 货号 | 407399 |
| 用途 | This product is for research use only, not for human or veterinary use. |
| 包装规格 | 5.0mg; 10.0mg; |
| CAS编号 | 1202580-59-3 |
| 纯度 | >98%% |
| 是否进口 | 是 |
Description: GPP78, also known as CAY10618, is a NMPRTase Inhibitor. The inhibition of NAD synthesis or salvage pathways has been proposed as a novel target for antitumoral drugs. GPP78 displays an IC(50) for cytotoxicity in vitro of 3.8 +/- 0.3 nM and an IC(50) for NAD depletion of 3.0 +/- 0.4 nM.
Synonym: GPP78; GPP-78; GPP 78; CAY10618; CAY-10618; CAY 10618.
IUPAC/Chemical Name: N-([1,1'-biphenyl]-2-yl)-8-(4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl)octanamide
InChi Key: SJOLTIOPWDLDEB-UHFFFAOYSA-N
InChi Code: InChI=1S/C27H29N5O/c33-27(29-25-16-9-8-15-24(25)22-12-5-4-6-13-22)17-7-2-1-3-10-19-32-21-26(30-31-32)23-14-11-18-28-20-23/h4-6,8-9,11-16,18,20-21H,1-3,7,10,17,19H2,(H,29,33)
SMILES Code: O=C(NC1=C(C2=CC=CC=C2)C=CC=C1)CCCCCCCN3N=NC(C4=CC=CN=C4)=C3
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: >2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
